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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 11 hits in this display   

TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50100871((Z)-1-(benzo[d]oxazol-2-yl)octadec-9-en-1-one | (Z...)
Affinity DataKi:  73nMAssay Description:Inhibition of human recombinant FAAHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50100871((Z)-1-(benzo[d]oxazol-2-yl)octadec-9-en-1-one | (Z...)
Affinity DataKi:  150nMAssay Description:Inhibitory activity against fatty acid amide hydrolase (FAAH)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50100871((Z)-1-(benzo[d]oxazol-2-yl)octadec-9-en-1-one | (Z...)
Affinity DataKi:  370nMAssay Description:Inhibition of rat FAAHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50100871((Z)-1-(benzo[d]oxazol-2-yl)octadec-9-en-1-one | (Z...)
Affinity DataKi:  370nMAssay Description:Inhibition of rat FAAH assessed as conversion [14]C-oleamide to oleic acidMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50100871((Z)-1-(benzo[d]oxazol-2-yl)octadec-9-en-1-one | (Z...)
Affinity DataKi:  370nMAssay Description:Inhibitory constant determined against recombinant Fatty-acid amide hydrolase from rat expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50100871((Z)-1-(benzo[d]oxazol-2-yl)octadec-9-en-1-one | (Z...)
Affinity DataKi:  370nMAssay Description:Inhibition of rat FAAH assessed as reduction in [14C]oleamide conversion to oleic acid by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Mus musculus (mouse))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50100871((Z)-1-(benzo[d]oxazol-2-yl)octadec-9-en-1-one | (Z...)
Affinity DataKi:  370nMAssay Description:Inhibitor affinity of the compound towards enzymes of class serine hydrolase was determined using biotin or fluorescent as radioligand (FP-biotin or ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase 1(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50100871((Z)-1-(benzo[d]oxazol-2-yl)octadec-9-en-1-one | (Z...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory concentration against Triacylglycerol hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50100871((Z)-1-(benzo[d]oxazol-2-yl)octadec-9-en-1-one | (Z...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory concentration of fatty acid amide hydrolase using FP-Rh radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase 1(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50100871((Z)-1-(benzo[d]oxazol-2-yl)octadec-9-en-1-one | (Z...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory concentration of triacylgylcerol hydrolase using FP-Rh radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50100871((Z)-1-(benzo[d]oxazol-2-yl)octadec-9-en-1-one | (Z...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory concentration against Fatty-acid amide hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed