Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50082065(CHEMBL3422516)
Affinity DataEC50:  222nMAssay Description:Agonist activity at human NPFF1R expressed in CHO cells assessed as effect on forskolin-induced cAMP accumulation after 15 mins by luminescence based...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Umr7247

Curated by ChEMBL
LigandPNGBDBM50082065(CHEMBL3422516)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed