Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50383315(CHEMBL2029773)
Affinity DataKi:  0.400nMpH: 5.0Assay Description:Competitive inhibition of wild type human glucocerebrosidase using 4-methylumbelliferyl beta-D-glucopyranoside as substrate after 15 mins by Dixon an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic beta-glucosidase(Homo sapiens (Human))
University Of British Columbia

Curated by ChEMBL
LigandPNGBDBM50383315(CHEMBL2029773)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human cytosolic beta-glucosidase using 4-methylumbelliferyl beta-D-glucopyranoside as substrate after 15 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed