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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetCytosolic phospholipase A2(Homo sapiens (Human))
University Of MüNster

Curated by ChEMBL
LigandPNGBDBM50185355(1-(3-(4-octylphenoxy)-2-oxopropyl)-1H-indole-5-car...)
Affinity DataIC50:  120nMAssay Description:Inhibition of human isolated cPLA2alpha by vescicle assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2(Homo sapiens (Human))
University Of MüNster

Curated by ChEMBL
LigandPNGBDBM50185355(1-(3-(4-octylphenoxy)-2-oxopropyl)-1H-indole-5-car...)
Affinity DataIC50:  120nMAssay Description:Inhibition of human platelet cPLA2-alpha assessed as arachidonic acid release by vesicle assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2(Homo sapiens (Human))
University Of MüNster

Curated by ChEMBL
LigandPNGBDBM50185355(1-(3-(4-octylphenoxy)-2-oxopropyl)-1H-indole-5-car...)
Affinity DataIC50:  120nMAssay Description:Inhibition of cPLA2 from human platelets by RP-HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2(Homo sapiens (Human))
University Of MüNster

Curated by ChEMBL
LigandPNGBDBM50185355(1-(3-(4-octylphenoxy)-2-oxopropyl)-1H-indole-5-car...)
Affinity DataIC50:  770nMAssay Description:Inhibition of cPLA2alpha activity assessed by A23187-induced arachidonic acid release in human plateletMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of M£Nster

Curated by ChEMBL
LigandPNGBDBM50185355(1-(3-(4-octylphenoxy)-2-oxopropyl)-1H-indole-5-car...)
Affinity DataIC50:  6.40E+3nMAssay Description:Inhibition of FAAH from rat brain microsomes by RP-HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed