Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetMuscarinic acetylcholine receptor M1(RAT)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50300559(3-hexyl-2-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl...)
Affinity DataKi:  1.10E+5nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor in Wistar rat brain cortex membrane after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50300559(3-hexyl-2-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl...)
Affinity DataIC50:  6.32E+5nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor in Wistar rat brain cortex membrane after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed