Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetMu-type opioid receptor(GUINEA PIG)
Eisai

Curated by ChEMBL
LigandPNGBDBM50010548(2-[2-(2-{2-[3-(4-Hydroxy-phenyl)-2-methylamino-pro...)
Affinity DataIC50:  6.60nMAssay Description:Evaluated for inhibitory activity against Opioid receptor mu 1 of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Eisai

Curated by ChEMBL
LigandPNGBDBM50010548(2-[2-(2-{2-[3-(4-Hydroxy-phenyl)-2-methylamino-pro...)
Affinity DataIC50:  20nMAssay Description:Evaluated for inhibitory activity against Opioid receptor kappa 1 of rabbit vas deferens (RVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Eisai

Curated by ChEMBL
LigandPNGBDBM50010548(2-[2-(2-{2-[3-(4-Hydroxy-phenyl)-2-methylamino-pro...)
Affinity DataIC50:  22nMAssay Description:Evaluated for inhibitory activity against Opioid receptor delta 1 of mouse vas deferens (MVD).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed