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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
6
hits in this display
Target
Muscarinic acetylcholine receptor M1
(RAT)
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50453786
(CHEMBL2092949)
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Affinity Data
IC50: 2.5nM
Assay Description:
Binding activity against muscarinic acetylcholine receptor M1 in rat brain, using [3H]OXO-M as the radioligand.
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Muscarinic acetylcholine receptor M1
(RAT)
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50453786
(CHEMBL2092949)
Copy SMILES
Copy InChI
Affinity Data
IC50: 3.70nM
Assay Description:
Binding activity against muscarinic acetylcholine receptor M1 in rat brain, using [3H]-Pz as the radioligand.
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Muscarinic acetylcholine receptor M1
(RAT)
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50033148
(3-(3-Hexyloxy-pyrazin-2-yl)-1-aza-bicyclo[2.2.2]oc...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 4.5nM
Assay Description:
Binding activity against muscarinic acetylcholine receptor M1 in rat brain, using [3H]OXO-M as the radioligand.
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Muscarinic acetylcholine receptor M1
(RAT)
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50033148
(3-(3-Hexyloxy-pyrazin-2-yl)-1-aza-bicyclo[2.2.2]oc...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 6nM
Assay Description:
Binding activity against muscarinic acetylcholine receptor M1 in rat brain, using [3H]-Pz as the radioligand.
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Muscarinic acetylcholine receptor M1
(RAT)
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50369037
(CHEMBL1788236)
Copy SMILES
Copy InChI
Affinity Data
IC50: 11nM
Assay Description:
Binding activity against muscarinic acetylcholine receptor M1 in rat brain, using [3H]-Pz as the radioligand.
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Muscarinic acetylcholine receptor M1
(RAT)
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50369037
(CHEMBL1788236)
Copy SMILES
Copy InChI
Affinity Data
IC50: 11nM
Assay Description:
Binding activity against muscarinic acetylcholine receptor M1 in rat brain, using [3H]-Pz as the radioligand.
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI