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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Eisai

Curated by ChEMBL
LigandPNGBDBM50047499(1-{2-Dimethylamino-6-[3-(5-methyl-4-phenyl-imidazo...)
Affinity DataIC50:  43nMAssay Description:Tested for inhibition against acyl coenzyme A:cholesterol acyltransferase from rabbit intestine microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Eisai

Curated by ChEMBL
LigandPNGBDBM50047499(1-{2-Dimethylamino-6-[3-(5-methyl-4-phenyl-imidazo...)
Affinity DataIC50:  43nMAssay Description:Inhibition against acyl coenzyme A:cholesterol acyltransferase derived from rabbit intestine microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Eisai

Curated by ChEMBL
LigandPNGBDBM50047499(1-{2-Dimethylamino-6-[3-(5-methyl-4-phenyl-imidazo...)
Affinity DataIC50:  110nMAssay Description:Inhibition against acyl coenzyme A:cholesterol acyltransferase derived from rabbit aorta homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Eisai

Curated by ChEMBL
LigandPNGBDBM50047499(1-{2-Dimethylamino-6-[3-(5-methyl-4-phenyl-imidazo...)
Affinity DataIC50:  110nMAssay Description:Tested for inhibition against acyl coenzyme A:cholesterol acyltransferase from rabbit aorta homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed