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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Sapienza University Of Rome

LigandPNGBDBM23002(N-[2-(5-hydroxy-1H-indol-3-yl)ethyl]-4-(7-pentylna...)
Affinity DataIC50: >1.00E+4nMAssay Description:The antagonistic effects of test compounds were evaluated using HEK293 cells stably overexpressing human TRPV1. Experiments were carried out by measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Sapienza University Of Rome

LigandPNGBDBM23002(N-[2-(5-hydroxy-1H-indol-3-yl)ethyl]-4-(7-pentylna...)
Affinity DataIC50:  5.00E+4nMpH: 9.0 T: 2°CAssay Description:The effect of the test compounds on the enzymatic hydrolysis of [14C]anandamide was evaluated by using membranes prepared from rat brain. [14C]Ethano...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed