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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227913(CHEMBL431965)
Affinity DataIC50:  9.54E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227913(CHEMBL431965)
Affinity DataIC50:  3.21E+4nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed