Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50016915(CHEMBL334465 | Dibutyl-[2-(naphthalen-1-yloxy)-eth...)
Affinity DataKi:  150nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 1A receptor of rat hippocampal tissue using [3H]OH-DPAT as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Medical College Of Virginia/Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50016915(CHEMBL334465 | Dibutyl-[2-(naphthalen-1-yloxy)-eth...)
Affinity DataKi:  2.68E+3nMAssay Description:Agonist activity to the human recombinant 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50016915(CHEMBL334465 | Dibutyl-[2-(naphthalen-1-yloxy)-eth...)
Affinity DataKi:  9.00E+3nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 1B receptor of rat striatal membrane homogenate using [3H]5-HT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rattus norvegicus (Rat))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50016915(CHEMBL334465 | Dibutyl-[2-(naphthalen-1-yloxy)-eth...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory activity against beta adrenergic receptor of rat frontal cortex homogenate using (1.0 nM) [3H]- dihydroalprenololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed