Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetAndrogen receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

LigandBDBM18532(6-(dibutylamino)-4-(trifluoromethyl)-1,2-dihydroqu...)Copy SMILESCopy InChI

Affinity DataKi:  222nM ΔG°:  -39.5kJ/mole IC50:  29.5nM EC50:  1.28E+3nMpH: 7.4 T: 2°CAssay Description:The compounds were evaluated in a transcriptional activation assay with hAR in a mammalian cell background (CV-1) as the primary in vitro assay. Rece...More data for this Ligand-Target Pair

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