Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetAdenosine receptor A1(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50199271(4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-pu...)
Affinity DataKi:  46nMAssay Description:Displacement of [125I]ABA from human adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50199271(4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-pu...)
Affinity DataKi:  2.26E+3nMAssay Description:Displacement of [125I]ZM241385 from human adenosine A2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed