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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetNeutrophil elastase(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398079(CHEMBL2182018)
Affinity DataKi:  1.30E+4nMAssay Description:Noncompetitive inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398079(CHEMBL2182018)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measured for 20 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398079(CHEMBL2182018)
Affinity DataIC50:  9.20E+4nMAssay Description:Inhibition of thrombin assessed as hydrolysis of H-D-Pro-L-Phe-L-Arg-p-nitroanilide incubated for 2 hrs measured for 20 mins by microplate reader ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398079(CHEMBL2182018)
Affinity DataIC50:  1.20E+5nMAssay Description:Inhibition of cathepsin G assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Phe-p-nitroanilide incubated for 2 hrs measured for 20 mins by microplate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed