Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50111694(5-Bromo-2-[(4-butoxy-benzenesulfonyl)-methyl-amino...)
Affinity DataIC50:  21nMAssay Description:Inhibition of Matrix metalloproteinase-9 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50111694(5-Bromo-2-[(4-butoxy-benzenesulfonyl)-methyl-amino...)
Affinity DataIC50:  21nMAssay Description:Inhibition of Matrix metalloproteinase-9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50111694(5-Bromo-2-[(4-butoxy-benzenesulfonyl)-methyl-amino...)
Affinity DataIC50:  67nMAssay Description:Inhibition of porcine Tumor necrosis factor alpha converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50111694(5-Bromo-2-[(4-butoxy-benzenesulfonyl)-methyl-amino...)
Affinity DataIC50:  67nMAssay Description:Inhibition of Tumor necrosis factor alpha converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50111694(5-Bromo-2-[(4-butoxy-benzenesulfonyl)-methyl-amino...)
Affinity DataIC50:  68nMAssay Description:Inhibition of Matrix metalloproteinase-13 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50111694(5-Bromo-2-[(4-butoxy-benzenesulfonyl)-methyl-amino...)
Affinity DataIC50:  68nMAssay Description:Inhibition of Matrix metalloproteinase-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50111694(5-Bromo-2-[(4-butoxy-benzenesulfonyl)-methyl-amino...)
Affinity DataIC50:  2.49E+3nMAssay Description:Inhibition of Matrix metalloproteinase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50111694(5-Bromo-2-[(4-butoxy-benzenesulfonyl)-methyl-amino...)
Affinity DataIC50:  2.49E+3nMAssay Description:Inhibition of Matrix metalloproteinase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed