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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 9 hits in this display   

TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50030732(CHEMBL323506 | N-{3-[3-Butyl-4-(3-fluoro-2'(tert-b...)
Affinity DataIC50:  0.170nMAssay Description:Inhibitory concentration of the compound against AT1 receptor from rat adrenal tissues.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50030732(CHEMBL323506 | N-{3-[3-Butyl-4-(3-fluoro-2'(tert-b...)
Affinity DataIC50:  0.240nMAssay Description:In vitro ability of the compound to inhibit the binding of radioligand 125I[Sar1,IIe8]AII to AT2 receptor from rat midbrainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50030732(CHEMBL323506 | N-{3-[3-Butyl-4-(3-fluoro-2'(tert-b...)
Affinity DataIC50:  0.240nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor, type 2 in rat midbrain membrane preparations.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50030732(CHEMBL323506 | N-{3-[3-Butyl-4-(3-fluoro-2'(tert-b...)
Affinity DataIC50:  0.700nMAssay Description:Inhibitory concentration against AT1 receptor from rat adrenal tissues.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50030732(CHEMBL323506 | N-{3-[3-Butyl-4-(3-fluoro-2'(tert-b...)
Affinity DataIC50:  0.820nMAssay Description:Inhibitory concentration of the compound against cloned human AT1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030732(CHEMBL323506 | N-{3-[3-Butyl-4-(3-fluoro-2'(tert-b...)
Affinity DataIC50:  0.840nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor, type 1 in rabbit aorta membrane preparations.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030732(CHEMBL323506 | N-{3-[3-Butyl-4-(3-fluoro-2'(tert-b...)
Affinity DataIC50:  0.840nMAssay Description:In vitro ability of the compound to inhibit the binding of radioligand 125I[Sar1,IIe8]AII to AT1 receptor from rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50030732(CHEMBL323506 | N-{3-[3-Butyl-4-(3-fluoro-2'(tert-b...)
Affinity DataIC50:  12nMAssay Description:In vitro inhibitory concentration of the compound against AT2 receptor from human adrenal tissues.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50030732(CHEMBL323506 | N-{3-[3-Butyl-4-(3-fluoro-2'(tert-b...)
Affinity DataIC50:  14nMAssay Description:In vitro inhibitory concentration of the compound against AT1 receptor from human adrenal tissues.More data for this Ligand-Target Pair
In DepthDetails Article