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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50039888(4'-[3-Butyl-1-(2-chloro-phenyl)-5-oxo-1,5-dihydro-...)
Affinity DataIC50:  1.40nMAssay Description:Displacement of 125I[Sar,Ile] from rabbit aorta membrane Angiotensin II receptor type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50039888(4'-[3-Butyl-1-(2-chloro-phenyl)-5-oxo-1,5-dihydro-...)
Affinity DataIC50:  1.40nMAssay Description:In vitro inhibitory activity against angiotensin II rabbit aorta AT1 receptor using radioligand [125I]-Sar Ile-AIIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(RAT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039888(4'-[3-Butyl-1-(2-chloro-phenyl)-5-oxo-1,5-dihydro-...)
Affinity DataIC50:  590nMAssay Description:In vitro inhibitory activity against angiotensin II rat midbrain AT2 receptor using radioligand [125I]-Sar Ile-AIIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed