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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetType-1 angiotensin II receptor(RABBIT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50044523(5-Butyl-2-cyclohexylmethyl-4-[2'-(2H-tetrazol-5-yl...)
Affinity DataIC50:  2.90nMAssay Description:In vitro antagonistic activity for angiotensin II receptor, type 1 by displacing 125I[Sar, ILe8 ]AII radioligand in rabbit aorta membrane without usi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50044523(5-Butyl-2-cyclohexylmethyl-4-[2'-(2H-tetrazol-5-yl...)
Affinity DataIC50:  2.90nMAssay Description:Antagonist activity at angiotensin 2 type-1 receptor in Oryctolagus cuniculus (rabbit) aorta in presence of bovine serum albuminMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50044523(5-Butyl-2-cyclohexylmethyl-4-[2'-(2H-tetrazol-5-yl...)
Affinity DataIC50:  2.90nMAssay Description:Antagonist activity at angiotensin 2 type-1 receptor in Oryctolagus cuniculus (rabbit) aorta in presence of bovine serum albuminMore data for this Ligand-Target Pair
In DepthDetails Article