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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
6
hits in this display
Target
Type-1 angiotensin II receptor
(RABBIT)
TBA
Ligand
BDBM50044346
(5-Butyl-2-propyl-4-[2'-(1H-tetrazol-5-yl)-biphenyl...)
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Affinity Data
IC50: 8.20nM
Assay Description:
Antagonist activity at angiotensin 2 type-1 receptor in Oryctolagus cuniculus (rabbit) aorta in presence of bovine serum albumin
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
Copy BDB DOI
Target
Type-1 angiotensin II receptor
(RABBIT)
TBA
Ligand
BDBM50044346
(5-Butyl-2-propyl-4-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 8.20nM
Assay Description:
In vitro antagonistic activity for angiotensin II receptor, type 1 by displacing 125I[Sar, ILe8 ]AII radioligand in rabbit aorta membrane without usi...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Type-1 angiotensin II receptor
(RABBIT)
TBA
Ligand
BDBM50044346
(5-Butyl-2-propyl-4-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 8.20nM
Assay Description:
Antagonist activity at angiotensin 2 type-1 receptor in Oryctolagus cuniculus (rabbit) aorta in presence of bovine serum albumin
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
Copy BDB DOI
Target
Type-1 angiotensin II receptor A/B
(RAT)
TBA
Ligand
BDBM50044346
(5-Butyl-2-propyl-4-[2'-(1H-tetrazol-5-yl)-biphenyl...)
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Affinity Data
IC50: 15nM
Assay Description:
Displacement of [125I]-angiotensin 2 from angiotensin AT1 receptor in Rattus norvegicus (rat) uterine membranes
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
Copy BDB DOI
Target
Type-1 angiotensin II receptor B
(RAT)
Searle R&D
Curated by
ChEMBL
Ligand
BDBM50044346
(5-Butyl-2-propyl-4-[2'-(1H-tetrazol-5-yl)-biphenyl...)
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Copy InChI
Affinity Data
IC50: 15nM
Assay Description:
Inhibition of [125I]-angiotensin-II binding to the angiotensin II receptor type 1 in rat uterine membranes
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Type-1 angiotensin II receptor A/B
(RAT)
TBA
Ligand
BDBM50044346
(5-Butyl-2-propyl-4-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 15nM
Assay Description:
Displacement of [125I]-angiotensin 2 from angiotensin AT1 receptor in Rattus norvegicus (rat) uterine membranes
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
Copy BDB DOI