Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetDipeptidase 1(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042555(5-Butyl-2-phenyl-4-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataKi:  5.90E+5nMAssay Description:In vitro apparent inhibition constant of porcine renal Dehydropeptidase-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042555(5-Butyl-2-phenyl-4-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50:  2.90nMAssay Description:Evaluation of Angiotensin II antagonistic activity by displacement of [125I]-Sar Ile-AII at the rabbit aorta Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Pseudomonas aeruginosa)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042555(5-Butyl-2-phenyl-4-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of metallo-beta-lactamase (MBL) from Pseudomonas aeruginosa mediated by the plasmid-borne IMP-1 enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase type 2(Bacteroides fragilis)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042555(5-Butyl-2-phenyl-4-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50:  2.00E+5nMAssay Description:Inhibition of metallo-beta-lactamase (MBL) from Bacteroides fragilis.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed