Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 9 hits in this display
BDBM50045861(2-(6H-Isoindolo[2,1-a]indol-11-yl)-N,N-dipropyl-ac...)
Ki: 20nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
BDBM50045861(2-(6H-Isoindolo[2,1-a]indol-11-yl)-N,N-dipropyl-ac...)
BDBM50045861(2-(6H-Isoindolo[2,1-a]indol-11-yl)-N,N-dipropyl-ac...)
IC50: >1.00E+3nMAssay Description:Inhibitory activity by measuring its ability to displace [125I]pindolol from beta-adrenergic receptor in rat brainMore data for this Ligand-Target Pair
BDBM50045861(2-(6H-Isoindolo[2,1-a]indol-11-yl)-N,N-dipropyl-ac...)
BDBM50045861(2-(6H-Isoindolo[2,1-a]indol-11-yl)-N,N-dipropyl-ac...)
BDBM50045861(2-(6H-Isoindolo[2,1-a]indol-11-yl)-N,N-dipropyl-ac...)
BDBM50045861(2-(6H-Isoindolo[2,1-a]indol-11-yl)-N,N-dipropyl-ac...)
BDBM50045861(2-(6H-Isoindolo[2,1-a]indol-11-yl)-N,N-dipropyl-ac...)
BDBM50045861(2-(6H-Isoindolo[2,1-a]indol-11-yl)-N,N-dipropyl-ac...)