Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 9 hits in this display   

TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045861(2-(6H-Isoindolo[2,1-a]indol-11-yl)-N,N-dipropyl-ac...)
Affinity DataKi:  20nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045861(2-(6H-Isoindolo[2,1-a]indol-11-yl)-N,N-dipropyl-ac...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory activity by measuring its ability to displace [3H]L-365,260 from cholecystokinin receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rattus norvegicus (Rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045861(2-(6H-Isoindolo[2,1-a]indol-11-yl)-N,N-dipropyl-ac...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory activity by measuring its ability to displace [125I]pindolol from beta-adrenergic receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50045861(2-(6H-Isoindolo[2,1-a]indol-11-yl)-N,N-dipropyl-ac...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of [3H]naxolone binding to opiate receptors in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50045861(2-(6H-Isoindolo[2,1-a]indol-11-yl)-N,N-dipropyl-ac...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]clonidine from alpha-adrenergic receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50045861(2-(6H-Isoindolo[2,1-a]indol-11-yl)-N,N-dipropyl-ac...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory activity by measuring its ability to displace [3H]WB-4101 from alpha-adrenergic receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A/1B/1D/1F(RAT)
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045861(2-(6H-Isoindolo[2,1-a]indol-11-yl)-N,N-dipropyl-ac...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory activity by measuring its ability to displace [3H]ketanserin from serotonin receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045861(2-(6H-Isoindolo[2,1-a]indol-11-yl)-N,N-dipropyl-ac...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory activity, measured by displacement [3H]-CP-55,940 from cannabinoid receptor (CB1) in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50045861(2-(6H-Isoindolo[2,1-a]indol-11-yl)-N,N-dipropyl-ac...)
Affinity DataIC50: >1.00E+3nMAssay Description:Tested for inhibitory activity by measuring its ability to displace [3H]3-PPP from opiate receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed