Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50001980(6-Dipropylamino-6,7-dihydro-5H-pyrido[1,2,3-de]qui...)
Affinity DataKi:  933nMAssay Description:Ability to displace [3H]-DPAT from 5-hydroxytryptamine 1A receptor in homogenates of bovine hippocampus.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50001980(6-Dipropylamino-6,7-dihydro-5H-pyrido[1,2,3-de]qui...)
Affinity DataKi: >1.00E+3nMAssay Description:Ability to displace [3H]raclopride from dopamine receptor D2 in rat striatal homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed