Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL

LigandBDBM50425097(CHEMBL2313230)Copy SMILESCopy InChI

Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human Kv1.5 channel expressed in CHO cells by high throughput planar patch clamp assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL

LigandBDBM50425097(CHEMBL2313230)Copy SMILESCopy InChI

Affinity DataIC50: >3.30E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProtUniProtKB/TrEMBL
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetIntermediate conductance calcium-activated potassium channel protein 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL

LigandBDBM50425097(CHEMBL2313230)Copy SMILESCopy InChI

Affinity DataIC50: >3.30E+4nMAssay Description:Inhibition of IK channel (unknown origin)More data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
DrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI