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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034323((2 beta-methyl) 8-Methoxy-2-methyl-1-propyl-2,3,3a...)
Affinity DataKi:  11nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034323((2 beta-methyl) 8-Methoxy-2-methyl-1-propyl-2,3,3a...)
Affinity DataKi:  11nMAssay Description:Binding affinity against [3H]8-OH-DPAT-labeled 5-hydroxytryptamine 1A receptor sites in bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034323((2 beta-methyl) 8-Methoxy-2-methyl-1-propyl-2,3,3a...)
Affinity DataKi:  11nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from bovine hippocampus, used [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50034323((2 beta-methyl) 8-Methoxy-2-methyl-1-propyl-2,3,3a...)
Affinity DataKi:  464nMAssay Description:Compound was tested for agonistic activity against D2 receptor from cloned CHO cells, used [3H]U-86170 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50034323((2 beta-methyl) 8-Methoxy-2-methyl-1-propyl-2,3,3a...)
Affinity DataKi:  464nMAssay Description:Binding affinity against [3H]U-86,170-labeled dopamine receptor D2 in cloned CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50034323((2 beta-methyl) 8-Methoxy-2-methyl-1-propyl-2,3,3a...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration against [3H]raclopride-labeled dopamine receptor D2 in rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed