Home
About
Info
Download
WebServices
Contact
Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Melatonin receptor type 1A
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM50117902
(CHEMBL3612606)
Copy SMILES
Copy InChI
Affinity Data
Ki: 5.80nM
Assay Description:
Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 mins
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melatonin receptor type 1A
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM50117902
(CHEMBL3612606)
Copy SMILES
Copy InChI
Affinity Data
EC50: 2nM
Assay Description:
Intrinsic activity at human MT1 receptor transfected in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI