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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 14 hits in this display   

Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50399616(CHEMBL2181188)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]GR113808 from human recombinant 5HT4R expressed in HEK293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50399616(CHEMBL2181188)
Affinity DataKi:  21.9nMAssay Description:Displacement of [3H]GR113808 from 5HT4R in guinea pig striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50399616(CHEMBL2181188)
Affinity DataKi:  98nMAssay Description:Binding affinity to human 5HT2B by Cerep protocol based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50399616(CHEMBL2181188)
Affinity DataKi:  729nMAssay Description:Binding affinity to human 5HT2C by Cerep protocol based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50399616(CHEMBL2181188)
Affinity DataKi:  1.78E+3nMAssay Description:Binding affinity to human 5HT2A by Cerep protocol based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50399616(CHEMBL2181188)
Affinity DataKi:  1.91E+3nMAssay Description:Binding affinity to human 5HT7 by Cerep protocol based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50399616(CHEMBL2181188)
Affinity DataKi:  2.36E+3nMAssay Description:Binding affinity to human 5HT1D by Cerep protocol based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50399616(CHEMBL2181188)
Affinity DataKi:  2.47E+3nMAssay Description:Binding affinity to human 5HT3 by Cerep protocol based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50399616(CHEMBL2181188)
Affinity DataKi:  6.26E+3nMAssay Description:Binding affinity to human 5HT6 by Cerep protocol based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50399616(CHEMBL2181188)
Affinity DataKi:  8.84E+3nMAssay Description:Binding affinity to human 5HT1A by Cerep protocol based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50399616(CHEMBL2181188)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human 5HT1B by Cerep protocol based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50399616(CHEMBL2181188)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human 5HT1E by Cerep protocol based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50399616(CHEMBL2181188)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human 5HT5A by Cerep protocol based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50399616(CHEMBL2181188)
Affinity DataEC50:  251nMAssay Description:Inverse agonist activity at human recombinant 5HT4R expressed in HEK293T cells assessed as Gs activationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed