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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetMelatonin receptor type 1B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50136404(1-[(S)-1-(2,3-Dihydro-benzofuran-4-yl)-pyrrolidin-...)
Affinity DataKi:  5.80nMAssay Description:Binding affinity against human MT2 melatonin receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50136404(1-[(S)-1-(2,3-Dihydro-benzofuran-4-yl)-pyrrolidin-...)
Affinity DataKi:  18nMAssay Description:Binding affinity against human MT1 melatonin receptor expressed in NIH3T3 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed