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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 10 hits in this display   

Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50005258(CHEMBL18762 | D-367 | [2-(4-Bromo-2,5-dimethoxy-ph...)
Affinity DataKi:  89nMAssay Description:Compound was tested for its ability to inhibit high affinity uptake of [3H]DA into rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50005258(CHEMBL18762 | D-367 | [2-(4-Bromo-2,5-dimethoxy-ph...)
Affinity DataKi:  514nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50005258(CHEMBL18762 | D-367 | [2-(4-Bromo-2,5-dimethoxy-ph...)
Affinity DataKi:  521nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50005258(CHEMBL18762 | D-367 | [2-(4-Bromo-2,5-dimethoxy-ph...)
Affinity DataKi:  976nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50005258(CHEMBL18762 | D-367 | [2-(4-Bromo-2,5-dimethoxy-ph...)
Affinity DataKi:  1.32E+3nMAssay Description:Evaluated for binding affinity towards rat cortical membranes at 5-hydroxytryptamine 1 receptor binding site by using [3H]-5-HT as a radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50005258(CHEMBL18762 | D-367 | [2-(4-Bromo-2,5-dimethoxy-ph...)
Affinity DataKi:  1.32E+3nMAssay Description:Binding affinity for 5-hydroxytryptamine 1 receptor of rat prefrontal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50005258(CHEMBL18762 | D-367 | [2-(4-Bromo-2,5-dimethoxy-ph...)
Affinity DataKi:  1.93E+3nMAssay Description:Displacement of [3H]ketanserin from rat prefrontal cortex 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50005258(CHEMBL18762 | D-367 | [2-(4-Bromo-2,5-dimethoxy-ph...)
Affinity DataKi:  1.93E+3nMAssay Description:Binding affinity to rat cortical membranes at 5-hydroxytryptamine 2 (5-HT2) receptor using [3H]KET as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50005258(CHEMBL18762 | D-367 | [2-(4-Bromo-2,5-dimethoxy-ph...)
Affinity DataKi:  2.46E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor from frontal cortical regions of male Sprague-Dawley rat homogenates, using [3H]ketanserin as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50005258(CHEMBL18762 | D-367 | [2-(4-Bromo-2,5-dimethoxy-ph...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1C receptor from frontal cortical regions of male Sprague-Dawley rat homogenates, using [3H]mesulergine ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed