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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hit in this display   

TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM139935(US8901087, 42)
Affinity DataKi:  1.03nM ΔG°:  -51.3kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
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