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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Mirati Therapeutics

US Patent
LigandPNGBDBM270466(US10059668, Example 29 | US10059668, Example 40)
Affinity DataIC50:  21nMpH: 7.5 T: 2°CAssay Description:Briefly, compounds of the present invention were solubilized in DMSO and a series of 10, three-fold serial dilutions were made for each compound in 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Mirati Therapeutics

US Patent
LigandPNGBDBM270466(US10059668, Example 29 | US10059668, Example 40)
Affinity DataIC50:  98nMpH: 7.5 T: 2°CAssay Description:Briefly, compounds of the present invention were solubilized in DMSO and a series of 10, three-fold serial dilutions were made for each compound in 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Mirati Therapeutics

US Patent
LigandPNGBDBM270466(US10059668, Example 29 | US10059668, Example 40)
Affinity DataIC50:  133nMpH: 7.5 T: 2°CAssay Description:Briefly, compounds of the present invention were solubilized in DMSO and a series of 10, three-fold serial dilutions were made for each compound in 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent