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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Alpha-2A adrenergic receptor
(BOVINE)
Merck Sharp And Dohme Research Laboratories
Curated by
ChEMBL
Ligand
BDBM50002147
(8-Piperazin-1-yl-3-propyl-imidazo[1,2-a]pyrazine; ...)
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Affinity Data
Ki: 480nM
Assay Description:
Binding affinity at Alpha-2 adrenergic receptor in calf cerebral cortex homogenates by [3H]clonidine displacement.
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Beta-2 adrenergic receptor
(GUINEA PIG)
Merck Sharp And Dohme Research Laboratories
Curated by
ChEMBL
Ligand
BDBM50002147
(8-Piperazin-1-yl-3-propyl-imidazo[1,2-a]pyrazine; ...)
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Copy InChI
Affinity Data
Ki: 1.39E+3nM
Assay Description:
Binding affinity against Beta-2 adrenergic receptor was measured using [125I]CYP as radioligand
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Beta-1 adrenergic receptor
(GUINEA PIG)
Merck Sharp And Dohme Research Laboratories
Curated by
ChEMBL
Ligand
BDBM50002147
(8-Piperazin-1-yl-3-propyl-imidazo[1,2-a]pyrazine; ...)
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Copy InChI
Affinity Data
Ki: 7.79E+3nM
Assay Description:
Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacement
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/TrEMBL
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI