Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 3 hits in this display
BDBM50159969(4-{3-[4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro...)
Ki: 207nMAssay Description:Binding affinity for adenosine A2b receptor by using as [3H]-ZM-241,385 (14 nM) radioligand in membranes from HEK-A2B cellsMore data for this Ligand-Target Pair
BDBM50159969(4-{3-[4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro...)
Ki: 288nMAssay Description:Binding affinity for adenosine A1 receptor by using as [3H]-CPX (0.5 nM) radioligand in membranes from Chinese hamster ovary cellsMore data for this Ligand-Target Pair
BDBM50159969(4-{3-[4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro...)
Ki: >5.00E+3nMAssay Description:Binding affinity for adenosine A2a receptor by using as [3H]-ZM-241,385 (2 nM) radioligand in membranes from HEK-A2A cellsMore data for this Ligand-Target Pair