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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetAdenosine receptor A1(GUINEA PIG)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50005390(1,3-Dipropyl-8-(1H-tetrazol-5-yl)-3,7-dihydro-puri...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against adenosine A1 receptor using N6-[3H]cyclohexyladenosine as radioligand in guinea pig forebrain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50005390(1,3-Dipropyl-8-(1H-tetrazol-5-yl)-3,7-dihydro-puri...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity against adenosine A2 receptor using N-[3H]-ethyladenosin-5''-uronamide as radioligand in rat striatal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed