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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Adenosine receptor A1
(Rattus norvegicus (rat))
Kyowa Hakko Kogyo
Curated by
ChEMBL
Ligand
BDBM50044431
(8-(Hexahydro-2,5-methano-pentalen-3a-yl)-1,3-dipro...)
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Affinity Data
Ki: 0.190nM
Assay Description:
Tested for binding affinity against Adenosine A1 receptor from rat forebrain membranes, using N6-[3H]- cyclohexyladenosine as radioligand
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
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Target
Adenosine receptor A1
(GUINEA PIG)
Kyowa Hakko Kogyo
Curated by
ChEMBL
Ligand
BDBM50044431
(8-(Hexahydro-2,5-methano-pentalen-3a-yl)-1,3-dipro...)
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Copy InChI
Affinity Data
Ki: 1.30nM
Assay Description:
Binding affinity against Adenosine A1 receptor from guinea pig forebrain membranes by N6-[3H]- cyclohexyladenosine displacement.
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Adenosine receptor A2a/A2b
(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by
ChEMBL
Ligand
BDBM50044431
(8-(Hexahydro-2,5-methano-pentalen-3a-yl)-1,3-dipro...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 380nM
Assay Description:
Binding affinity at Adenosine A2 receptor from rat striatal membranes by N-[3H] ethyladenosin-5'- uronamide displacement.
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI