Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018716(2-Amino-N-[1-({[(1,3-dimethyl-butyl)-ethyl-carbamo...)
Affinity DataKi:  36nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018716(2-Amino-N-[1-({[(1,3-dimethyl-butyl)-ethyl-carbamo...)
Affinity DataKi:  3.45E+3nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50018716(2-Amino-N-[1-({[(1,3-dimethyl-butyl)-ethyl-carbamo...)
Affinity DataIC50:  216nMAssay Description:Inhibition of electrically evoked contraction of guinea pig ileum (myenteric plexus:longitudinal muscle preparation) by antagonist action at mu 1 opi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed