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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
6
hits in this display
Target
3-oxo-5-alpha-steroid 4-dehydrogenase 2
(Homo sapiens (Human))
TBA
Curated by
ChEMBL
Ligand
BDBM50213061
(CHEMBL2298601)
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Affinity Data
Ki: 2nM
Assay Description:
Inhibition of type-2 human steroid 5-alpha-reductase.
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
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Target
3-oxo-5-alpha-steroid 4-dehydrogenase 1
(Homo sapiens (Human))
TBA
Curated by
ChEMBL
Ligand
BDBM50213061
(CHEMBL2298601)
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Copy InChI
Affinity Data
Ki: 3nM
Assay Description:
Inhibition of type-1 human steroid 5-alpha-reductase
More data for this Ligand-Target Pair
Target Info
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
Copy BDB DOI
Target
3-oxo-5-alpha-steroid 4-dehydrogenase 1/2
(Rattus norvegicus)
TBA
Curated by
ChEMBL
Ligand
BDBM50213061
(CHEMBL2298601)
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Affinity Data
Ki: 5nM
Assay Description:
Apparent inhibitory constant value for rat prostatic steroid 5alpha reductase was determined
More data for this Ligand-Target Pair
Target Info
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
3-oxo-5-alpha-steroid 4-dehydrogenase 2
(Homo sapiens (Human))
TBA
Curated by
ChEMBL
Ligand
BDBM50213061
(CHEMBL2298601)
Copy SMILES
Copy InChI
Affinity Data
IC50: 8.60nM
Assay Description:
Inhibitory activity of the compound against human prostatic Steroid 5-alpha-reductase
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
Copy BDB DOI
Target
3-oxo-5-alpha-steroid 4-dehydrogenase 1/2
(Rattus norvegicus)
TBA
Curated by
ChEMBL
Ligand
BDBM50213061
(CHEMBL2298601)
Copy SMILES
Copy InChI
Affinity Data
IC50: 11nM
Assay Description:
In vitro inhibitory activity against rat prostatic steroid 5-alpha-reductase
More data for this Ligand-Target Pair
Target Info
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Androgen receptor
(Rattus norvegicus (Rat))
TBA
Curated by
ChEMBL
Ligand
BDBM50213061
(CHEMBL2298601)
Copy SMILES
Copy InChI
Affinity Data
IC50: 2.80E+3nM
Assay Description:
In vitro antagonist activity against rat prostatic androgen receptor (AR)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI