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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetAcetylcholinesterase(Rattus norvegicus (rat))
Sichuan University

LigandPNGBDBM167912(N,N-diethylcarbamic acid-4-(5-hydroxy-6,7-dimethox...)
Affinity DataIC50:  570nMAssay Description:For rat AChE or BuChE inhibition assays, a reaction mixture (100 μL) containing acetylthiocholine iodide (1 mmol/L, 30 μL) (J&K Scientific)...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Sichuan University

LigandPNGBDBM167912(N,N-diethylcarbamic acid-4-(5-hydroxy-6,7-dimethox...)
Affinity DataIC50:  570nMAssay Description:Inhibition of rat cortex AChE using acetylthiocholine iodide as substrate after 15 mins by Ellman methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Sichuan University

LigandPNGBDBM167912(N,N-diethylcarbamic acid-4-(5-hydroxy-6,7-dimethox...)
Affinity DataIC50:  570nMAssay Description:Inhibition of rat cortex AChE using acetylthiocholine iodide as substrate incubated for 15 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCarboxylic ester hydrolase(Rattus norvegicus (rat))
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM167912(N,N-diethylcarbamic acid-4-(5-hydroxy-6,7-dimethox...)
Affinity DataIC50:  2.26E+4nMAssay Description:Inhibition of rat serum BChE using butyrylthiocholine iodide as substrate incubated for 15 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCarboxylic ester hydrolase(Rattus norvegicus (rat))
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM167912(N,N-diethylcarbamic acid-4-(5-hydroxy-6,7-dimethox...)
Affinity DataIC50:  2.26E+4nMAssay Description:For rat AChE or BuChE inhibition assays, a reaction mixture (100 μL) containing acetylthiocholine iodide (1 mmol/L, 30 μL) (J&K Scientific)...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed