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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetB1 bradykinin receptor(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50308988((R)-N-(1-(1-(4-(diethylcarbamoyl)phenyl)ethylcarba...)
Affinity DataIC50:  3.10E+3nMAssay Description:Antagonist activity at bradikinin B1 receptor in human IMR90 cells assessed as inhibition of des-Arg-bradykinin-mediated calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed