Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 3 hits in this display
BDBM50077059(4-[((1R,2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-yl...)
BDBM50077059(4-[((1R,2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-yl...)
BDBM50077059(4-[((1R,2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-yl...)
IC50: 8.60E+3nMAssay Description:Binding affinity towards Opioid receptor kappa 1 using [3H]- U-69,593 (1.5 nM) as radioligand in guinea pig brain membranesMore data for this Ligand-Target Pair