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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Melanocortin receptor 4
(Homo sapiens (Human))
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50177564
(CHEMBL380540 | N-((R)-3-(4-chlorophenyl)-1-(4-(2-(...)
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Affinity Data
Ki: 5.80nM
Assay Description:
Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
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Target
Melanocortin receptor 5
(Homo sapiens (Human))
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50177564
(CHEMBL380540 | N-((R)-3-(4-chlorophenyl)-1-(4-(2-(...)
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Copy InChI
Affinity Data
Ki: 420nM
Assay Description:
Displacement of [125I]NDP-alpha-MSH from cloned human MC5R expressed in HEK293 cell
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanocortin receptor 3
(Homo sapiens (Human))
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50177564
(CHEMBL380540 | N-((R)-3-(4-chlorophenyl)-1-(4-(2-(...)
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Affinity Data
Ki: 1.90E+3nM
Assay Description:
Displacement of [125I]NDP-alpha-MSH from cloned human MC3R expressed in HEK293 cell
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanocyte-stimulating hormone receptor
(Homo sapiens (Human))
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50177564
(CHEMBL380540 | N-((R)-3-(4-chlorophenyl)-1-(4-(2-(...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 7.00E+3nM
Assay Description:
Displacement of [125I]NDP-alpha-MSH from cloned human MC1R expressed in HEK293 cell
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI