Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetPlatelet-activating factor acetylhydrolase(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50125262(CHEMBL10532 | N-(2-Diethylamino-ethyl)-2-[2-(4-flu...)
Affinity DataIC50:  1nMAssay Description:Inhibitory activity against recombinant human Lp-PLA2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50125262(CHEMBL10532 | N-(2-Diethylamino-ethyl)-2-[2-(4-flu...)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibitory activity against CYP450 3A4 isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50125262(CHEMBL10532 | N-(2-Diethylamino-ethyl)-2-[2-(4-flu...)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibitory activity against Cytochrome P450 2D6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed