Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetAdenosine receptor A2a(Homo sapiens (Human))
Panjab University

LigandPNGBDBM175378(8-[3-{2-(Diethylaminoethylamino)-2-oxoethoxy}-phen...)
Affinity DataKi:  179nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Panjab University

LigandPNGBDBM175378(8-[3-{2-(Diethylaminoethylamino)-2-oxoethoxy}-phen...)
Affinity DataKi:  1.22E+3nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Panjab University

LigandPNGBDBM175378(8-[3-{2-(Diethylaminoethylamino)-2-oxoethoxy}-phen...)
Affinity DataKi:  4.91E+3nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3 [I248L](Homo sapiens (Human))
Panjab University

LigandPNGBDBM175378(8-[3-{2-(Diethylaminoethylamino)-2-oxoethoxy}-phen...)
Affinity DataKi:  8.39E+3nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed