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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Muscarinic acetylcholine receptor M2
(RAT)
Institute Of Research
Curated by
ChEMBL
Ligand
BDBM50018230
(2-(4-Methylcarbamoyloxy-phenyl)-2-phenyl-propionic...)
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Affinity Data
Ki: 2nM
Assay Description:
Binding affinity was determined from the inhibition of contraction of guinea pig ileum which has Muscarinic acetylcholine receptor M2 subtype.
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Muscarinic receptor M1
(Bos taurus)
Institute Of Research
Curated by
ChEMBL
Ligand
BDBM50018230
(2-(4-Methylcarbamoyloxy-phenyl)-2-phenyl-propionic...)
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Affinity Data
Ki: 26nM
Assay Description:
Inhibition of [3H]NMS binding to cerebral cortex membranes which contain predominantly the Muscarinic acetylcholine receptor M1 subtypes
More data for this Ligand-Target Pair
Target Info
KEGG
UniProtKB/TrEMBL
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Cholinesterase
(Homo sapiens (Human))
Institute Of Research
Curated by
ChEMBL
Ligand
BDBM50018230
(2-(4-Methylcarbamoyloxy-phenyl)-2-phenyl-propionic...)
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Affinity Data
Ki: 1.40E+3nM
Assay Description:
Anticholinesterase activity by their ability to inactivate human serum butyrylcholinesterase
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI