Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 19 hits in this display
BDBM50005685(2,2-Diphenyl-propionic acid 2-diethylamino-ethyl e...)
BDBM50005685(2,2-Diphenyl-propionic acid 2-diethylamino-ethyl e...)
Ki: 1.70nMAssay Description:Inhibition of carbachol-induced release of alpha-amylase from pancreatic acinar cells from that of rat ileum contained the M2 receptor subtypesMore data for this Ligand-Target Pair
BDBM50005685(2,2-Diphenyl-propionic acid 2-diethylamino-ethyl e...)
BDBM50005685(2,2-Diphenyl-propionic acid 2-diethylamino-ethyl e...)
BDBM50005685(2,2-Diphenyl-propionic acid 2-diethylamino-ethyl e...)
BDBM50005685(2,2-Diphenyl-propionic acid 2-diethylamino-ethyl e...)
BDBM50005685(2,2-Diphenyl-propionic acid 2-diethylamino-ethyl e...)
BDBM50005685(2,2-Diphenyl-propionic acid 2-diethylamino-ethyl e...)
BDBM50005685(2,2-Diphenyl-propionic acid 2-diethylamino-ethyl e...)
BDBM50005685(2,2-Diphenyl-propionic acid 2-diethylamino-ethyl e...)
BDBM50005685(2,2-Diphenyl-propionic acid 2-diethylamino-ethyl e...)
Ki: 15.1nMAssay Description:Displacement of [3H] N-methylscopolamine from human muscarinic M1 receptor expressed in CHOK1 cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
BDBM50005685(2,2-Diphenyl-propionic acid 2-diethylamino-ethyl e...)
Ki: 23nMAssay Description:Inhibit the binding of [N-mnethyl-3H]-scopolamine [3H]-NMS) to Muscarinic acetylcholine receptor of human IRM-30 neuroblastoma cellsMore data for this Ligand-Target Pair
BDBM50005685(2,2-Diphenyl-propionic acid 2-diethylamino-ethyl e...)
Ki: 26.5nMAssay Description:Displacement of [3H] N-methylscopolamine from human muscarinic M1 receptor after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
BDBM50005685(2,2-Diphenyl-propionic acid 2-diethylamino-ethyl e...)
Ki: 51nMAssay Description:Inhibition of [3H]NMS binding to cerebral cortex membranes which contain predominantly the Muscarinic acetylcholine receptor M1 subtypesMore data for this Ligand-Target Pair
BDBM50005685(2,2-Diphenyl-propionic acid 2-diethylamino-ethyl e...)
Ki: 107nMAssay Description:Displacement of [3H] N-methylscopolamine from human muscarinic M2 receptor expressed in CHOK1 cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
BDBM50005685(2,2-Diphenyl-propionic acid 2-diethylamino-ethyl e...)
Ki: 628nMAssay Description:Displacement of [3H] N-methylscopolamine from human muscarinic M4 receptor expressed in CHOK1 cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
BDBM50005685(2,2-Diphenyl-propionic acid 2-diethylamino-ethyl e...)
Ki: 7.76E+3nMAssay Description:Displacement of [3H] N-methylscopolamine from human muscarinic M3 receptor expressed in CHOK1 cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
BDBM50005685(2,2-Diphenyl-propionic acid 2-diethylamino-ethyl e...)
BDBM50005685(2,2-Diphenyl-propionic acid 2-diethylamino-ethyl e...)