Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase/7-dehydrocholesterol reductase(Homo sapiens (Human))
University Of Georgia

Curated by ChEMBL

LigandBDBM50020286(4-{1-Chloro-2-[4-(2-diethylamino-ethoxy)-phenyl]-2...)Copy SMILESCopy InChI

Affinity DataIC50:  32nMAssay Description:Displacement of [3H]tamoxifen from antiestrogen binding site (AEBS)More data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
DrugBankantibodypediaantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetEstrogen receptor beta(Homo sapiens (Human))
University Of Georgia

Curated by ChEMBL

LigandBDBM50020286(4-{1-Chloro-2-[4-(2-diethylamino-ethoxy)-phenyl]-2...)Copy SMILESCopy InChI

Affinity DataIC50:  3.00E+3nMAssay Description:Displacement of [3H]-estradiol from estrogen receptor (ER)More data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI