Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091350(CHEMBL3582270)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1B adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091350(CHEMBL3582270)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1A adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091350(CHEMBL3582270)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1D adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091350(CHEMBL3582270)
Affinity DataIC50:  0.600nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1A adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091350(CHEMBL3582270)
Affinity DataIC50:  1.20nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1B adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50091350(CHEMBL3582270)
Affinity DataIC50:  2.20nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1D adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed