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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Oxysterols receptor LXR-alpha
(Homo sapiens (Human))
F. Hoffmann-La Roche
Curated by
ChEMBL
Ligand
BDBM50192137
(2-(3-chloro-4-(((2-(3-chlorophenyl)-5-methyloxazol...)
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Affinity Data
IC50: 2nM
Assay Description:
Binding affinity to LXRalpha by radioligand displacement assay
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Oxysterols receptor LXR-beta
(Homo sapiens (Human))
F. Hoffmann-La Roche
Curated by
ChEMBL
Ligand
BDBM50192137
(2-(3-chloro-4-(((2-(3-chlorophenyl)-5-methyloxazol...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 4nM
Assay Description:
Binding affinity to LXRbeta by radioligand displacement assay
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Oxysterols receptor LXR-beta
(Homo sapiens (Human))
F. Hoffmann-La Roche
Curated by
ChEMBL
Ligand
BDBM50192137
(2-(3-chloro-4-(((2-(3-chlorophenyl)-5-methyloxazol...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 40nM
Assay Description:
Transactivation of LXRbeta by luciferase reporter gene assay
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Oxysterols receptor LXR-alpha
(Homo sapiens (Human))
F. Hoffmann-La Roche
Curated by
ChEMBL
Ligand
BDBM50192137
(2-(3-chloro-4-(((2-(3-chlorophenyl)-5-methyloxazol...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 300nM
Assay Description:
Transactivation of LXRalpha by luciferase reporter gene assay
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI