Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetMuscarinic acetylcholine receptor M1(RAT)
Institute For Drug Discovery Research

Curated by ChEMBL
LigandPNGBDBM50044702(3-Ethyl-8-methyl-2-thioxo-1-oxa-3,8-diaza-spiro[4....)
Affinity DataKi:  890nMAssay Description:Displacement of [3H]pirenzepine from rat cortex membrane expressing muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Institute For Drug Discovery Research

Curated by ChEMBL
LigandPNGBDBM50044702(3-Ethyl-8-methyl-2-thioxo-1-oxa-3,8-diaza-spiro[4....)
Affinity DataKi:  4.30E+3nMAssay Description:Compound tested in vitro for displacement of [3H]quinuclidinyl benzilate from rat cerebellum membrane expressing muscarinic M2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed