Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetAdenosine receptor A3(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50454476(CHEMBL2113630)
Affinity DataKi:  6.60nMAssay Description:Displacement of [125I]AB-MECA from cloned rat Adenosine A3 receptor in stably transfected CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50454476(CHEMBL2113630)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50454476(CHEMBL2113630)
Affinity DataKi:  3.36E+3nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2A receptor in rat striatal homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed