Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetAdenosine receptor A1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50202570(1-deoxy-1-{6-[N'-(furan-2-carbonyl)-hydrazino]-9H-...)
Affinity DataKi:  1.05E+3nMAssay Description:Displacement of [3H]CHA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50202570(1-deoxy-1-{6-[N'-(furan-2-carbonyl)-hydrazino]-9H-...)
Affinity DataKi:  1.55E+3nMAssay Description:Displacement of [3H]CGS-21680 from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50202570(1-deoxy-1-{6-[N'-(furan-2-carbonyl)-hydrazino]-9H-...)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50202570(1-deoxy-1-{6-[N'-(furan-2-carbonyl)-hydrazino]-9H-...)
Affinity DataEC50:  82nMAssay Description:Activity at human adenosine A2B receptor expressed in CHO cells assessed as stimulation of cAMP levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50202570(1-deoxy-1-{6-[N'-(furan-2-carbonyl)-hydrazino]-9H-...)
Affinity DataEC50:  1.22E+7nMAssay Description:Agonist activity at human adenosine A2B receptor expressed in CHO cells assessed as stimulation of adenylate cyclaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed